发明名称 |
NOVEL ARYLAMIDINE DERIVATIVE OR SALT THEREOF |
摘要 |
An arylamidine derivative represented by a general formula described below or a salt thereof has an excellent antifungal action and high safety, and it is useful as an antifungal agent with good pharmacokinetics and pharmacodynamic properties: (see above formula) wherein X represents an unsubstituted or substituted lower alkylene or alkenylene group; G1 represents an oxygen atom, a sulfur atom, or an imino group; G2 represents a carbon atom or a nitrogen atom; R a represents at least one group selected from the group consisting of a hydrogen atom, a halogen atom, and unsubstituted or substituted alkyl, cycloalkyl and alkoxy groups; R1 represents an unprotected or protected or unsubstituted or substituted amidino group; and R2 represents a substituted amino or substituted cyclic amino group, or the like.
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申请公布号 |
CA2477212(C) |
申请公布日期 |
2011.11.15 |
申请号 |
CA20032477212 |
申请日期 |
2003.03.04 |
申请人 |
TOYAMA CHEMICAL CO., LTD. |
发明人 |
HAYASHI, KAZUYA;OJIMA, KATSUJI;HORI, KOZO;OKUJO, NORIYUKI;MITSUYAMA, JUNICHI;KUNITANI, KAZUTO;TOHDO, KEISUKE |
分类号 |
C07D295/088;A61K31/138;A61K31/44;A61K31/445;A61K31/495;A61P31/10;C07C257/18;C07C259/18;C07C271/64;C07C323/62;C07D207/14;C07D211/22;C07D211/26;C07D211/58;C07D213/62;C07D213/78;C07D213/85;C07D241/04;C07D241/08;C07D243/08;C07D245/02;C07D261/12;C07D295/092;C07D295/13;C07D401/06;C07D413/06 |
主分类号 |
C07D295/088 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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