发明名称 METHOD FOR PREPARING TETRAZOLE METHANESULFONIC ACID SALTS, AND NOVEL COMPOUND USED IN SAME
摘要 According to the present invention, a method for preparing tetrazole methanesulfonic acid salts comprises an acylation reaction using a novel 4-iodine-4H-chromene-2-carbothionic acid S-benzothiazole-2-yl ester. The method of the present invention can shorten a reaction time and improve safety as compared to conventional methods, and can prepare high-purity tetrazole methanesulfonic acid salts at a high yield rate without using a column chromatography method.
申请公布号 WO2011087316(A3) 申请公布日期 2011.11.10
申请号 WO2011KR00291 申请日期 2011.01.14
申请人 HANMI HOLDINGS CO., LTD.;BANG, KEUK CHAN;PARK, BUM WOO;CHOI, JONG WON;LEE, JAE CHUL;AN, YONG HOON;AHN, YOUNG GIL;KIM, MAENG SUP 发明人 BANG, KEUK CHAN;PARK, BUM WOO;CHOI, JONG WON;LEE, JAE CHUL;AN, YONG HOON;AHN, YOUNG GIL;KIM, MAENG SUP
分类号 C07D405/14;C07D403/02;C07D417/12 主分类号 C07D405/14
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