发明名称 PYRAZOLYL QUINAZOLINE KINASE INHIBITORS
摘要 The invention relates to new quinoxaline derivative compounds, to pharmaceutical compositions comprising said compounds, to processes for the preparation of said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
申请公布号 WO2011135376(A1) 申请公布日期 2011.11.03
申请号 WO2011GB50851 申请日期 2011.04.28
申请人 ASTEX THERAPEUTICS LIMITED;SAXTY, GORDON;MURRAY, CHRISTOPHER WILLIAM;BERDINI, VALERIO;BESONG, GILBERT EBAI;HAMLETT, CHRISTOPHER CHARLES FREDERICK;JOHNSON, CHRISTOPHER NORBERT;WOODHEAD, STEVEN JOHN;READER, MICHAEL;REES, DAVID CHARLES;MEVELLEC, LAURENCE ANNE;ANGIBAUD, PATRICK RENE;FREYNE, EDDY JEAN EDGARD;GOVAERTS, TOM CORNELIS HORTENSE;WEERTS, JOHAN ERWIN EDMOND;PERERA, TIMOTHY PIETRO SUREN;GILISSEN, RONALDUS ARNODUS HENDRIKA JOSEPH;WROBLOWSKI, BERTHOLD;LACRAMPE, JEAN FERNAND ARMAND;PAPANIKOS, ALEXANDRA;QUEROLLE, OLIVER ALEXIS GEORGES;PASQUIER, ELISABETH THERESE JEANNE;PILATTE, ISABELLE NOELLE CONSTANCE;BONNET, PASCAL GHISLAIN ANDRE;EMBRECHTS, WERNER CONSTANT JOHAN;AKKARI, RHALID;MEERPOEL, LIEVEN 发明人 SAXTY, GORDON;MURRAY, CHRISTOPHER WILLIAM;BERDINI, VALERIO;BESONG, GILBERT EBAI;HAMLETT, CHRISTOPHER CHARLES FREDERICK;JOHNSON, CHRISTOPHER NORBERT;WOODHEAD, STEVEN JOHN;READER, MICHAEL;REES, DAVID CHARLES;MEVELLEC, LAURENCE ANNE;ANGIBAUD, PATRICK RENE;FREYNE, EDDY JEAN EDGARD;GOVAERTS, TOM CORNELIS HORTENSE;WEERTS, JOHAN ERWIN EDMOND;PERERA, TIMOTHY PIETRO SUREN;GILISSEN, RONALDUS ARNODUS HENDRIKA JOSEPH;WROBLOWSKI, BERTHOLD;LACRAMPE, JEAN FERNAND ARMAND;PAPANIKOS, ALEXANDRA;QUEROLLE, OLIVER ALEXIS GEORGES;PASQUIER, ELISABETH THERESE JEANNE;PILATTE, ISABELLE NOELLE CONSTANCE;BONNET, PASCAL GHISLAIN ANDRE;EMBRECHTS, WERNER CONSTANT JOHAN;AKKARI, RHALID;MEERPOEL, LIEVEN
分类号 C07D403/04;A61K31/498;A61P35/00;C07D403/14;C07D405/14;C07D409/14;C07D413/14;C07D487/08 主分类号 C07D403/04
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