发明名称 NAPHTHRIDINE DERIVATIVES AS PI3K INHIBITORS FOR THE TREATMENT OF CANCER AND IMMUNE - INFLAMMATORY DISEASES
摘要 <p>Compounds of formulae (I) and (II): or a pharmaceutically acceptable salt thereof, wherein: R1 is a nitrogen-containing 5 to 7-membered heteroaryl or heterocycle; R2 and R3 are each independently (LQ)mY, are described. The compounds are PI3K inhibitors and are useful for the treatment of cancer and immune-inflammatory diseases.</p>
申请公布号 WO2011135351(A1) 申请公布日期 2011.11.03
申请号 WO2011GB50824 申请日期 2011.04.26
申请人 KARUS THERAPEUTICS LIMITED;SHUTTLEWORTH, STEPHEN, JOSEPH;SILVA, FRANCK, ALEXANDRE 发明人 SHUTTLEWORTH, STEPHEN, JOSEPH;SILVA, FRANCK, ALEXANDRE
分类号 C07D471/04;A61K31/4375;A61P29/00;A61P35/00;A61P37/00 主分类号 C07D471/04
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