发明名称 |
CRYSTALLINE POLYMORPHS OF A CXC-CHEMOKINE RECEPTOR LIGAND. |
摘要 |
THE PRESENT INVENTION RELATES TO FOUR DISTINCT CRYSTALLINE POLYMORPHS OF A MONOHYDRATE OF COMPOUND A HAVING THE FOLLOWING CHEMICAL STRUCTURE: THESE FOUR POLYMORPHIC FORMS, HEREIN REFERRED TO AS FORMS I, II, III AND IV ARE ACTIVE AS A CXC-CHEMOKINE RECEPTOR LIGANDS. THE INVENTION IS FURTHER DIRECTED TO FORMULATIONS, METHODS OF TREATMENT, AND PROCESSES OF SYNTHESIS OF THESE POLYMORPHIC FORMS.
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申请公布号 |
MY144657(A) |
申请公布日期 |
2011.10.31 |
申请号 |
MYPI20050328 |
申请日期 |
2005.01.28 |
申请人 |
SCHERING CORPORATION |
发明人 |
HU, MENGWEI;KLOPFER, KEVIN;YU, YOUNONG;DWYER, MICHAEL;TAVERAS, ARTHUR G.;KIN-MEADE, AGNES;YIN, JIANGUO;FU, XIAOYONG;MCALLISTER, TIMOTHY;ZHANG, SHUYI |
分类号 |
A61K31/341;A61K31/34;C07D307/52 |
主分类号 |
A61K31/341 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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