发明名称 BETA-CARBOLINES AS INHIBITORS OF HASPIN AND DYRK KINASES
摘要 The present disclosure is directed to compounds of Formula ( I ) which are inhibitors of Haspin kinase and DYRK kinases. The compounds of the present disclosure, and compositions thereof, are useful in the treatment of disease related to Haspin kinase and DYRK kinase expression and/or activity.
申请公布号 WO2011133795(A2) 申请公布日期 2011.10.27
申请号 WO2011US33466 申请日期 2011.04.21
申请人 THE BRIGHAM AND WOMEN'S HOSPITAL, INC.;HIGGINS, JONATHAN;PATNAIK, DEBASIS;ULYANOVA, NATALIA;STEIN, ROSS L.;XIAN, JUN;GLICKSMAN, MARCIE;CUNY, GREGORY D. 发明人 HIGGINS, JONATHAN;PATNAIK, DEBASIS;ULYANOVA, NATALIA;STEIN, ROSS L.;XIAN, JUN;GLICKSMAN, MARCIE;CUNY, GREGORY D.
分类号 C07D471/04;A61K31/403;A61K31/437;A61P3/10;A61P35/00;C07D209/88;C07D491/147 主分类号 C07D471/04
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