发明名称 |
NOVEL HETEROCYCLIC COMPOUNDS FOR USE AS METAP-2 INHIBITORS |
摘要 |
<p>Compounds of the formula I, in which D, X, Y, Z, R and R1 have the meanings indicated in Claim 1, are inhibitors of methionine aminopeptidase and can be employed for the treatment of tumors.</p> |
申请公布号 |
EP2379558(A1) |
申请公布日期 |
2011.10.26 |
申请号 |
EP20090796971 |
申请日期 |
2009.12.22 |
申请人 |
MERCK PATENT GMBH |
发明人 |
HEINRICH, TIMO;ZENKE, FRANK;KRIER, MIREILLE;SCHIEMANN, KAI |
分类号 |
C07D487/04;A61K31/519;A61P35/00 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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