发明名称 |
INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY AND USE THEREOF TO TREAT OPHTHALMIC DISORDERS |
摘要 |
<p>Disclosed are compounds, and compositions of same, that are protein tyrosine kinase inhibitors. The compounds find use in the treatment of ophthalmic diseases, disorders and conditions. Said compounds are of the formulae (I), (II) or (III). Wherein R = (IV), (V), (VI), (VII), (VIII), (IX), (X), (XI) or (XII).</p> |
申请公布号 |
WO2011127565(A1) |
申请公布日期 |
2011.10.20 |
申请号 |
WO2011CA00390 |
申请日期 |
2011.04.08 |
申请人 |
METHYLGENE INC.;OTSUKA PHARMACEUTICAL CO. LTD;RAEPPEL, STEPHANE;ZHAN, LIJIE;CLARIDGE, STEPHEN WILLIAM;RAEPPEL, FRANCK;GAUDETTE, FREDERIC;VAISBURG, ARKADII |
发明人 |
RAEPPEL, STEPHANE;ZHAN, LIJIE;CLARIDGE, STEPHEN WILLIAM;RAEPPEL, FRANCK;GAUDETTE, FREDERIC;VAISBURG, ARKADII |
分类号 |
C07D495/04;A61K31/4365;A61K31/444;A61K31/496;A61K31/5377;A61P27/02 |
主分类号 |
C07D495/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|