发明名称 METHOD OF PREPARING SITAGLIPTIN AND INTERMEDIATES USED THEREIN
摘要 Disclosed are a novel, simple and low-cost method for preparing sitagliptin, as DPP-IV (dipeptidyl peptidase IV) inhibitor, which is useful in treating type 2 diabetes mellitus and key intermediates used in said preparation of sitagliptin.
申请公布号 WO2011049344(A3) 申请公布日期 2011.10.13
申请号 WO2010KR07150 申请日期 2010.10.19
申请人 HANMI HOLDINGS CO., LTD.;KIM, NAM DU;CHANG, JI YEON;KIM, DONG JUN;LEE, HYUN SEUNG;JUNG, JAE HYUK;CHANG, YOUNG KIL;LEE, GWAN SUN 发明人 KIM, NAM DU;CHANG, JI YEON;KIM, DONG JUN;LEE, HYUN SEUNG;JUNG, JAE HYUK;CHANG, YOUNG KIL;LEE, GWAN SUN
分类号 C07D487/04;A61K31/4985;A61P3/10;C07D487/02 主分类号 C07D487/04
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