发明名称 Arylethynyl derivatives
摘要 The present invention relates to ethynyl compounds of formula I wherein R1, R2, R2′, R3, R3′, R4, R4′, U, V, W, Y, m, and n are as defined herein and to a pharmaceutically acceptable acid addition salts, to a racemic mixtures, or to its corresponding enantiomers and/or optical isomers and/or stereoisomers thereof. Compounds of formula I are allosteric modulators of the metabotropic glutamate receptor subtype 5 (mGluR5).
申请公布号 US2011251169(A1) 申请公布日期 2011.10.13
申请号 US201113066044 申请日期 2011.04.05
申请人 GREEN LUKE;GUBA WOLFGANG;JAESCHKE GEORG;JOLIDON SYNESE;LINDEMANN LOTHAR;RICCI ANTONIO;RUEHER DANIEL;STADLER HEINZ;VIEIRA ERIC 发明人 GREEN LUKE;GUBA WOLFGANG;JAESCHKE GEORG;JOLIDON SYNESE;LINDEMANN LOTHAR;RICCI ANTONIO;RUEHER DANIEL;STADLER HEINZ;VIEIRA ERIC
分类号 A61K31/397;A61K31/4439;A61K31/444;A61K31/501;A61K31/506;A61K31/5355;A61K31/5377;A61K31/541;A61P25/28;C07D401/04;C07D401/14;C07D403/04;C07D413/04;C07D417/04 主分类号 A61K31/397
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