发明名称 NOVEL INTERMEDIATE AND PROCESS FOR PREPARING ENTECAVIR USING SAME
摘要 The present invention relates to a novel, high-yield and low-cost method for preparing entecavir, [1-S-(1α,3α,4&bgr;)]-2-amino-1,9-dihydro-9-[4-hydroxy-3-(hydroxymethyl)-2-methylenecyclopentyl]-6H-purin-6-one, an antiviral agent, and novel intermediates used therein.
申请公布号 US2011251387(A1) 申请公布日期 2011.10.13
申请号 US200913140640 申请日期 2009.12.24
申请人 HANMI HOLDINGS CO., LTD. 发明人 LEE JAEHEON;PARK GHA-SEUNG;KIM JIN HEE;LEE JI EUN;PARK CHUL HYUN;CHOI TAE JIN;PARK EUN-JU;KIM CHEOL KYUNG;LIM EUN JUNG;CHANG YOUNG-KIL;LEE GWAN SUN
分类号 C07D473/18;C07C49/517;C07F7/08 主分类号 C07D473/18
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