发明名称 |
PROCESS FOR THE PRODUCTION OF BIVALIRUDIN |
摘要 |
The present invention relates to a process for the production of bivalirudin, a 20-mer peptide of formula H-D-Phe1-Pro-Arg-Pro-Gly5-Gly-Gly-Gly-Asn-Gly10-Asp-Phe-Glu-Glu-Ile14-Pro-Glu-Glu-Tyr-Lee-OH (I) via a convergent five-fragment synthesis, and to several peptide intermediates thereof.
|
申请公布号 |
US2011251372(A1) |
申请公布日期 |
2011.10.13 |
申请号 |
US200913139956 |
申请日期 |
2009.12.17 |
申请人 |
SOMMEN GEOFFROY;FORNI LUCIANO |
发明人 |
SOMMEN GEOFFROY;FORNI LUCIANO |
分类号 |
C07K7/08;C07K1/107;C07K5/107;C07K7/06 |
主分类号 |
C07K7/08 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|