发明名称 PROCESS FOR THE PRODUCTION OF BIVALIRUDIN
摘要 The present invention relates to a process for the production of bivalirudin, a 20-mer peptide of formula H-D-Phe1-Pro-Arg-Pro-Gly5-Gly-Gly-Gly-Asn-Gly10-Asp-Phe-Glu-Glu-Ile14-Pro-Glu-Glu-Tyr-Lee-OH (I) via a convergent five-fragment synthesis, and to several peptide intermediates thereof.
申请公布号 US2011251372(A1) 申请公布日期 2011.10.13
申请号 US200913139956 申请日期 2009.12.17
申请人 SOMMEN GEOFFROY;FORNI LUCIANO 发明人 SOMMEN GEOFFROY;FORNI LUCIANO
分类号 C07K7/08;C07K1/107;C07K5/107;C07K7/06 主分类号 C07K7/08
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