发明名称 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS
摘要 The present invention relates to a compounds of formula I wherein A, Ar1, Ar2, R1, R2, R3, R4, R5, R6, m, n, o, p, s, t, and u are as defined herein or to a pharmaceutically active salt, a racemic mixture, an enantiomer, an optical isomer or a tautomeric form thereof. the present compounds are high potential NK-3 receptor antagonists for the treatment of depression, pain, psychosis, Parkinson's disease, schizophrenia, anxiety and attention deficit hyperactivity disorder (ADHD).
申请公布号 KR20110111312(A) 申请公布日期 2011.10.10
申请号 KR20117019521 申请日期 2010.01.19
申请人 F. HOFFMANN-LA ROCHE AG 发明人 KNUST HENNER;NETTEKOVEN MATTHIAS;RATNI HASANE;RIEMER CLAUS;VIFIAN WALTER
分类号 C07D413/14;A61K31/4545;A61P25/00;C07D401/14 主分类号 C07D413/14
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