发明名称 Process for preparing pyridinamines and novel polymorphs thereof
摘要 Disclosed herein are crystalline polymorph form II of 3-chloro-N-(3-chloro-5-trifluoromethyl-2-pyridy)-á,á,á-trifluoro-2,6dinitro-p-toluidine (fluazinam) exhibiting at least one of the following characteristics: a) an X-ray powder diffraction pattern having characteristic peaks expressed in degrees 2è (+/-0.2°è) at about 7.4, 10.4, 13.4, 15.1, 18.95, 20, 20.4, 21.05, 21.3, 22.2, 24.9, 27.15, 28.6 and 30.5; b) a predominant endotherm at about 109°C as measured by a Differential Scanning Calorimeter (DSC) at a scan rate of 10°C per minute. Also disclosed are processes for the preparation of crystalline polymorphs above, compositions comprising said polymorphs and uses thereof. The compositions are useful in combating insects, mites, fungus and bacteria.
申请公布号 NZ567671(A) 申请公布日期 2011.09.30
申请号 NZ20060567671 申请日期 2006.11.23
申请人 MAKHTESHIM CHEMICAL WORKS LTD 发明人 COHEN, SHLOMI;ZAMIR, SHARONA
分类号 A61K31/44;A01N43/40;C07D213/74;C07D213/85 主分类号 A61K31/44
代理机构 代理人
主权项
地址