发明名称 CRYSTALLINE SOLVATES AND COMPLEXES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL) METHYL) PHENYL)-D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 Disclosed is a crystalline structure of a (1S)-1,5-anhydro-1-C-(3-((phenyl) methyl) phenyl)-D-glucitol of formula 1c. Also disclosed is the use of said form for treating diabetes, insulin resistance, hyperglycemia, hyperinsulinemia, elevated blood levels of fatty acids or glycerol, hyperlipidemia, dyslipidemia, obesity, hypertriglyceridemia, or diabetic complications.
申请公布号 NZ589190(A) 申请公布日期 2011.09.30
申请号 NZ20070589190 申请日期 2007.06.21
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 GOUGOUTAS, JACK Z;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT P;BIEN, JEFFREY T;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETEROF;GROSSO, JOHN ANTHONY;NIRSCHL, ALEXANDRA A;SINGH, JANAK;DIMARCO, JOHN D (DECEASED, REPRESENTED BY DORIS DIMARCO)
分类号 C07H7/04;A61K31/70;A61P3/10 主分类号 C07H7/04
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