发明名称 SOLID FORMS OF (R)-1(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL)-N-(1-(2,3-DIHYDEROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2-YL)-1H-INDOL-5-YL) CYCLOPROPANECARBOXAMIDE
摘要 The present invention relates to solid forms of (R)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2- methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide (Compound 1) in substantially crystalline form (Form A) or amorphous form, pharmaceutical compositions thereof, and methods of treatment therewith.
申请公布号 WO2011119984(A1) 申请公布日期 2011.09.29
申请号 WO2011US30032 申请日期 2011.03.25
申请人 VERTEX PHARMACEUTICALS INCORPORATED;KESHAVARZ-SHOKRI, ALI;ZHANG, BEILI;ALCACIO, TIM, EDWARD;LEE, ELAINE, CHUNGMIN;ZHANG, YUEGANG;KRAWIEC, MARIUSZ 发明人 KESHAVARZ-SHOKRI, ALI;ZHANG, BEILI;ALCACIO, TIM, EDWARD;LEE, ELAINE, CHUNGMIN;ZHANG, YUEGANG;KRAWIEC, MARIUSZ
分类号 C07D405/12;A61K31/404;A61P11/00 主分类号 C07D405/12
代理机构 代理人
主权项
地址