发明名称 MOLECULAR CRYSTAL OF (4 -(1,8-NAPHTHYRIDIN-2-YL) PIPERIDIN - 1 -YL ) PYRIMIDINE DERIVATIVE
摘要 <p>A molecular crystal form of (S)-3-(2,5-dimethyl-6-(4-(5,6,7,8-tetrahydro-1,8- naphthyridin-2-yl)piperidin- 1 -yl)pyrimidin-4-ylamino)-2-(4- methoxyphenylsulfonamido)propanoic acid is characterized by an X-ray powder diffraction ("XRPD") spectrum that comprises peaks at 2? angles of 7.44, 14.80, 16.64, and 23.04 ±0.2°. The molecular crystal can be formulated into pharmaceutical composition for treating or controlling diseases resulting from pathological angiogenesis.</p>
申请公布号 WO2011119282(A1) 申请公布日期 2011.09.29
申请号 WO2011US25865 申请日期 2011.02.23
申请人 BAUSCH & LOMB INCORPORATED;PHILLIPS, ERIC;SHAWER, MOHANNAD 发明人 PHILLIPS, ERIC;SHAWER, MOHANNAD
分类号 C07D471/04;A61K31/506 主分类号 C07D471/04
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