发明名称 BICYCLIC PEPTIDOMIMETIC INHIBITORS OF ASPARTYL-PROTEASES FOR THE TREATMENT OF INFECTIOUS DISEASES
摘要 The present invention refers to 3-aza-bicyclo[3.2.1]octane derivatives of general formula (I) their preparation, use and pharmaceutical compositions useful in the treatment of pathologies associated with microbial pathogens expressing aspartyl-protease activity.
申请公布号 US2011237577(A1) 申请公布日期 2011.09.29
申请号 US200913130666 申请日期 2009.11.24
申请人 CASSONE ANTONIO;DE BERNARDIS FLAVIA;GARACI ENRICO;TRABOCCHI ANDREA;GUARNA ANTONIO 发明人 CASSONE ANTONIO;DE BERNARDIS FLAVIA;GARACI ENRICO;TRABOCCHI ANDREA;GUARNA ANTONIO
分类号 A61K31/5386;A61P31/00;A61P31/10;A61P31/14;A61P31/18;A61P33/02;C07D498/08 主分类号 A61K31/5386
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