发明名称 |
BICYCLIC PEPTIDOMIMETIC INHIBITORS OF ASPARTYL-PROTEASES FOR THE TREATMENT OF INFECTIOUS DISEASES |
摘要 |
The present invention refers to 3-aza-bicyclo[3.2.1]octane derivatives of general formula (I) their preparation, use and pharmaceutical compositions useful in the treatment of pathologies associated with microbial pathogens expressing aspartyl-protease activity.
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申请公布号 |
US2011237577(A1) |
申请公布日期 |
2011.09.29 |
申请号 |
US200913130666 |
申请日期 |
2009.11.24 |
申请人 |
CASSONE ANTONIO;DE BERNARDIS FLAVIA;GARACI ENRICO;TRABOCCHI ANDREA;GUARNA ANTONIO |
发明人 |
CASSONE ANTONIO;DE BERNARDIS FLAVIA;GARACI ENRICO;TRABOCCHI ANDREA;GUARNA ANTONIO |
分类号 |
A61K31/5386;A61P31/00;A61P31/10;A61P31/14;A61P31/18;A61P33/02;C07D498/08 |
主分类号 |
A61K31/5386 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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