发明名称 AN IMPROVED PROCESS FOR THE PREPARATION OF AMLODIPINE FREE BASE AND ACID ADDITION SALTS THEREOF
摘要 <p>Disclosed herein is an improved process for preparation of Amlodipine free base and acid addition salts thereof in good yield by deprotecting Phthaloyl Amlodipine using total concentration of 25% aqueous monomethyl amine in the reaction mixture and Amlodipine free base thus obtained is treated with suitable acids in aqueous medium to yield corresponding Amlodipine salts.</p>
申请公布号 WO2011117876(A1) 申请公布日期 2011.09.29
申请号 WO2010IN00296 申请日期 2010.05.06
申请人 FDC LIMITED;CHANDAVARKAR, MOHAN, ANAND;SOHANI, SUHAS, VASANT;BHOIR, VIJTKUMAR, GAJANAN;SAWANT, SAMEER, NARAYAN 发明人 CHANDAVARKAR, MOHAN, ANAND;SOHANI, SUHAS, VASANT;BHOIR, VIJTKUMAR, GAJANAN;SAWANT, SAMEER, NARAYAN
分类号 C07D211/82;C07D401/12 主分类号 C07D211/82
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