发明名称 SUBSTITUTED PYRAZOLE DERIVATIVE
摘要 <p>Disclosed are a novel pyrazole derivative and an androgen receptor antagonist containing the pyrazole derivative. Specifically disclosed is a compound represented by the formula (I') below or a salt thereof. (In the formula, R1 represents a hydrogen atom, a group having a carbon atom serving as a bonding hand, a group having a nitrogen atom serving as a bonding hand, a group having an oxygen atom serving as a bonding hand or a group having a sulfur atom serving as a bonding hand; R2 represents a phenyl group having a cyano (which may further have a substituent other than cyano); R3 represents a hydrogen atom, a group having a carbon atom serving as a bonding hand, a group having a nitrogen atom serving as a bonding hand, a group having an oxygen atom serving as a bonding hand or a group having a sulfur atom serving as a bonding hand; R4 represents an optionally substituted cyclic group; and X represents an optionally substituted methylene or CO.)</p>
申请公布号 TN2010000091(A1) 申请公布日期 2011.09.26
申请号 TN20100000091 申请日期 2010.02.23
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED 发明人 ITO MITSUHIRO;SUZAKI TOMOHIKO;YAMAMOTO SATOSHI
分类号 A61K31/415;A61K31/4162;A61K31/4178;A61K31/4196;A61K31/42;C07D231/12 主分类号 A61K31/415
代理机构 代理人
主权项
地址