发明名称 |
2,3 DIHYDRO-1H-INDEN-1-YL-2,7-DIAZASPIRO [3.5] NONANE DERIVATIVES AND THEIR USE AS ANTAGONISTS OR INVERSE AGONISTS OF THE GHRELIN RECEPTOR |
摘要 |
The present invention provides a compound of Formula (I) or a pharmaceutically salt thereof wherein R1, R2, Ra, L, Z, Z1 and Z2 are as defined herein, that act as Ghrelin antagonists or inverse agonists; pharmaceutical compositions thereof; and methods of treating diseases, disorders, or conditions mediated by the antagonism of the Ghrelin receptor. |
申请公布号 |
CA2792234(A1) |
申请公布日期 |
2011.09.22 |
申请号 |
CA20112792234 |
申请日期 |
2011.03.11 |
申请人 |
PFIZER INC. |
发明人 |
BHATTACHARYA, SAMIT KUMAR;CAMERON, KIMBERLY O'KEEFE;FERNANDO, DILINIE PRASADHINI;KUNG, DANIEL WEI-SHUNG;LONDREGAN, ALLYN TIMOTHY;MCCLURE, KIM FRANCIS;SIMILA, SUVI TUULA MARJUKKA |
分类号 |
C07D471/10;A61K31/4747;A61P3/04;A61P3/10;C07D519/00 |
主分类号 |
C07D471/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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