发明名称 |
PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS |
摘要 |
Methods of treating an SCD-mediated disease or condition in a mammal, preferably a human, are disclosed, wherein the methods comprise administering to a mammal in need thereof a compound of formula (Ia): where x, y, W, V, R2, R3, R4, R5, R6, R6a, R7, R7a, R8, R8a, R9 and R9a are defined herein. Pharmaceutical compositions comprising the compounds of formula (I) are also disclosed.
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申请公布号 |
CA2597069(C) |
申请公布日期 |
2011.09.20 |
申请号 |
CA20062597069 |
申请日期 |
2006.02.08 |
申请人 |
XENON PHARMACEUTICALS INC. |
发明人 |
ABREO, MELWYN;HOLLADAY, MARK W.;LI, WENBAO;SUN, SENGEN;TU, CHI;GSCHWEND, HEINZ W.;CHAFEEV, MIKHAIL;CHAKKA, NAGASREE;CHOWDHURY, SULTAN;FU, JIAN-MIN;HOU, DUANJIE;KAMBOJ, RAJENDER;KODUMURU, VISHNUMURTHY;LIU, SHIFENG;RAINA, VANDNA;SUN, SHAOYI;SVIRIDOV, SERGUEI;WINTHER, MICHAEL D.;ZHANG, ZAIHUL |
分类号 |
C07D237/20;A61K31/00;A61K31/501;A61K31/551;A61P3/06;C07D237/22;C07D237/24 |
主分类号 |
C07D237/20 |
代理机构 |
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地址 |
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