发明名称 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS |
摘要 |
The present invention provides heteroaryl substituted pyrrolo[2,3-b]pyridines and heteroaryl substituted pyrrolo[2,3-b]pyrimidines that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases, skin disorders, myeloid proliferative disorders, cancer, and other diseases. |
申请公布号 |
US2011223210(A1) |
申请公布日期 |
2011.09.15 |
申请号 |
US201113076220 |
申请日期 |
2011.03.30 |
申请人 |
INCYTE CORPORATION, A DELAWARE CORPORATION |
发明人 |
RODGERS JAMES D.;SHEPARD STACEY;MADUSKUIE, JR. THOMAS P.;WANG HAISHENG;FALAHATPISHEH NIKOO;RAFALSKI MARIA;ARVANITIS ARGYRIOS G.;STORACE LOUIS;JALLURI RAVIKUMAR;FRIDMAN JORDAN S.;VADDI KRISHNA |
分类号 |
A61K31/519;A61K9/00;A61P7/00;A61P35/00;A61P35/02;A61P43/00 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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