发明名称 |
BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS |
摘要 |
The invention provides compounds of the formula (I): The compounds have activity against cyclin dependent kinases, glycogen synthase kinase and Aurora kinases and are therefore useful to treat cancer and viral diseases. |
申请公布号 |
US2011224203(A1) |
申请公布日期 |
2011.09.15 |
申请号 |
US201113116121 |
申请日期 |
2011.05.26 |
申请人 |
ASTEX THERAPEUTICS LIMITED |
发明人 |
BERDINI VALERIO;O'BRIEN MICHAEL ALISTAIR;CARR MARIA GRAZIA;EARLY THERESA RACHEL;NAVARRO EVA FIGUEROA;GILL ADRIAN LIAM;HOWARD STEVEN;TREWARTHA GARY;WOOLFORD ALISON JO-ANNE;WOODHEAD ANDREW JAMES;WYATT PAUL GRAHAM |
分类号 |
A61K31/5377;A61K31/00;A61K31/4184;A61P31/10;A61P35/00;A61P35/02;A61P35/04;C07D401/14;C07D405/14;C07D409/14;C07D413/14 |
主分类号 |
A61K31/5377 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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