PROCESS FOR THE PREPARATION OF 4-(3-CHLORO-2-FLUORO-ANILINO)-7-METHOXY-6-[1-(N-METHYLCARBAMOYLMETHYL)-PIPERIDIN-4-YL]QUINAZOLINE
摘要
Processes for the preparation of 4-(3-chloro-2-fluoroanilino)-7-methoxy-6-{[1-(N- methylcarbamoylmethyl)piperidin-4-yl]oxy}quinazoline, salts thereof, and the intermediates used in the process are described.
申请公布号
WO2010122340(A3)
申请公布日期
2011.09.09
申请号
WO2010GB50653
申请日期
2010.04.22
申请人
ASTRAZENECA AB;ASTRAZENECA UK LIMITED;BOARDMAN, KAY, ALISON;CUNNINGHAM, OLIVER, ROBERT;GOUNDRY, WILLIAM;LAFFAN, DAVID, DERMOT, PATRICK
发明人
BOARDMAN, KAY, ALISON;CUNNINGHAM, OLIVER, ROBERT;GOUNDRY, WILLIAM;LAFFAN, DAVID, DERMOT, PATRICK