发明名称 PROCESS FOR THE PREPARATION OF 4-(3-CHLORO-2-FLUORO-ANILINO)-7-METHOXY-6-[1-(N-METHYLCARBAMOYLMETHYL)-PIPERIDIN-4-YL]QUINAZOLINE
摘要 Processes for the preparation of 4-(3-chloro-2-fluoroanilino)-7-methoxy-6-{[1-(N- methylcarbamoylmethyl)piperidin-4-yl]oxy}quinazoline, salts thereof, and the intermediates used in the process are described.
申请公布号 WO2010122340(A3) 申请公布日期 2011.09.09
申请号 WO2010GB50653 申请日期 2010.04.22
申请人 ASTRAZENECA AB;ASTRAZENECA UK LIMITED;BOARDMAN, KAY, ALISON;CUNNINGHAM, OLIVER, ROBERT;GOUNDRY, WILLIAM;LAFFAN, DAVID, DERMOT, PATRICK 发明人 BOARDMAN, KAY, ALISON;CUNNINGHAM, OLIVER, ROBERT;GOUNDRY, WILLIAM;LAFFAN, DAVID, DERMOT, PATRICK
分类号 C07D211/46;C07C257/12;C07D401/12 主分类号 C07D211/46
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