发明名称 ARYL CARBOXAMIDE DERIVATIVES AS SODIUM CHANNEL INHIBITORS FOR TREATMENT OF PAIN
摘要 The present invention provides compounds that are inhibitors of voltage-gated sodium channels (Nav), in particular Nav 1.7, and are therefore useful for the treatment of diseases treatable by inhibition of these channels, in particular, chronic pain disorders. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.
申请公布号 WO2011103196(A1) 申请公布日期 2011.08.25
申请号 WO2011US25092 申请日期 2011.02.16
申请人 AMGEN INC.;BREGMAN, HOWARD;BUCHANAN, JOHN, L.;CHAKKA, NAGASREE;DIMAURO, ERIN, F.;DU, BINGFAN;NGUYEN, HANH, NHO;ZHENG, XIAO, MEI 发明人 BREGMAN, HOWARD;BUCHANAN, JOHN, L.;CHAKKA, NAGASREE;DIMAURO, ERIN, F.;DU, BINGFAN;NGUYEN, HANH, NHO;ZHENG, XIAO, MEI
分类号 C07D213/74;A61K31/4427;A61K31/505;A61K31/506;A61K31/53;A61P29/00;C07D239/48;C07D251/48;C07D401/04;C07D403/04;C07D471/10 主分类号 C07D213/74
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