发明名称 8-CARBOXAMIDO-2,6-METHANO-3-BENZAZOCINES
摘要 8-Substituted-2,6-methano-3-benzazocines of general structure I in which A is —CH2—OH, —CH2NH2, —NHSO2CH3, and Y is O, S or NOH are useful as analgesics, anti-diarrheal agents, anticonvulsants, antitussives and anti-addiction medications. 8-Carboxamides, thiocarboxamides, hydroxyamidines and formamides are preferred.
申请公布号 US2011207763(A1) 申请公布日期 2011.08.25
申请号 US201113103599 申请日期 2011.05.09
申请人 RENSSELAER POLYTECHNIC INSTITUTE 发明人 WENTLAND MARK P.
分类号 A61K31/485;A61K31/439;A61K31/4748;A61P1/00;A61P1/06;A61P1/12;A61P3/00;A61P3/04;A61P9/10;A61P11/00;A61P11/14;A61P13/02;A61P17/04;A61P25/00;A61P25/02;A61P25/04;A61P25/08;A61P25/28;A61P25/30;A61P25/36;A61P29/00;A61P37/06;A61P43/00;C07B61/00;C07D221/22;C07D221/26;C07D401/04;C07D405/06;C07D489/00;C07D489/08;C07D489/09;C07D489/10;C07D491/20;C07D491/22 主分类号 A61K31/485
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