发明名称 TRICYCLIC HETEROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF
摘要 The invention provides novel compounds of formula I having the general formula: wherein R1, R2, R3, X and Y are as described herein. Accordingly, the compounds may be provided in pharmaceutically acceptable compositions and used for the treatment of immunological or hyperproliferative disorders.
申请公布号 US2011201593(A1) 申请公布日期 2011.08.18
申请号 US201113004808 申请日期 2011.01.11
申请人 GENENTECH, INC. 发明人 BABU SRINIVASAN;BERGERON PHILLIPPE;DRAGOVICH PETER;DYKE HAZEL JOAN;GIBBONS PAUL;GRADL STEFAN;HANAN EMILY;HURLEY CHRISTOPHER;JOHNSON TONY;KOEHLER MICHAEL;KULAGOWSKI JANUSZ;LABADIE SHARADA;LYSSIKATOS JOSEPH;MENDONCA ROHAN;PULK REBECCA;WARD STUART;WASZKOWYCZ BOHDAN;ZAK MARK
分类号 A61K31/397;A61K31/437;A61K31/496;A61K31/506;A61K31/5377;A61K31/55;A61P11/06;A61P17/06;A61P19/02;A61P37/06;C07D413/14;C07D471/14 主分类号 A61K31/397
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