发明名称 CARBONIC ANHYDRASE INHIBITORS
摘要 A carbonic anhydrase IX (CA IX) inhibitor which comprises a compound of general formula: R-NH-CX-NH-(CH2)n-Ar-Q-SO2-NH2 or a pharmaceutically-acceptable salt, derivative or prodrug thereof; wherein n = 0, 1 or 2; Q is O or NH; X is O or S; and R comprises an organic substituent group.
申请公布号 WO2011098610(A1) 申请公布日期 2011.08.18
申请号 WO2011EP52156 申请日期 2011.02.14
申请人 UNIVERSITA DEGLI STUDI DI FIRENZE;UNIVERSITETET I OLSO;UNIVERSITY OF MANCHESTER;EBBESEN, PETER;SUPURAN, CLAUDIU T.;SCOZZAFAVA, ANDREA;PETTERSEN, ERIK OLAI;WILLIAMS, KAYE;PASTOREKOVA, SILVIA;DUBOIS, LUDWIG;LAMBIN, PHILIPPE 发明人 EBBESEN, PETER;SUPURAN, CLAUDIU T.;SCOZZAFAVA, ANDREA;PETTERSEN, ERIK OLAI;WILLIAMS, KAYE;PASTOREKOVA, SILVIA;DUBOIS, LUDWIG;LAMBIN, PHILIPPE
分类号 A61K31/18;A61P35/00;C07C311/00 主分类号 A61K31/18
代理机构 代理人
主权项
地址