发明名称 SALT FORMS OF 4-(4-METHYLPIPERAZIN-1-YLMETHYL)-N-[4-METHYL-3-(4-PYRIDIN-3-YL)PYRIMIDIN-2-YLAMINO)PHENYL]-BENZAMIDE.
摘要 THE PRESENT INVENTION RELATES TO ACID ADDITION SALTS OF 4-[(4-METHYL-1-PIPERAZINYL)METHYL]-N-(4- METHYL-3-[[4-(3-PYRIDINYL)-2-PYRIMIDINYL]AMINO]PHENYL]-BENZAMIDE, WHICH ARE SELECTED FROM THE GROUP CONSISTING OF A TARTRATE SALT, SUCH AS A (D)(-) TARTRATE SALT OR A (LJ(+) TARTRATE SALT, A HYDROCHLORIDE SALT, A CITRATE SALT, A MALATE SALT, A FUMARATE SALT, A SUCCINATE SALT, A BENZOATE SALT, A BENZENESULFONATE SALT, A PAMOATE SALT, A FORMATE SALT, A MALONATE SALT, A 1,5- NAPHTHALENEDISULFONATE SALT, A SALICYLATE SALT, A CYCLOHEXANESULFAMATE SALT, A LACTATE SALT, A MANDELATE SALT, AQ GLUTARATE SALT, AN ADIPATE SALT, A SQUARATE SALT, A VANILLATE SALT, AN OXALOACETATE SALT, AN ASCORBATE SALT AND A SULFATE SALT.
申请公布号 MY144177(A) 申请公布日期 2011.08.15
申请号 MY2005PI00400 申请日期 2005.02.02
申请人 NOVARTIS AG 发明人 HANS MICHAEL B0XDCRGER;PAUL WILLIAM MANLEY;MICHAEL MUTZ
分类号 C07D401/04 主分类号 C07D401/04
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