摘要 |
THE PRESENT INVENTION RELATES TO ACID ADDITION SALTS OF 4-[(4-METHYL-1-PIPERAZINYL)METHYL]-N-(4- METHYL-3-[[4-(3-PYRIDINYL)-2-PYRIMIDINYL]AMINO]PHENYL]-BENZAMIDE, WHICH ARE SELECTED FROM THE GROUP CONSISTING OF A TARTRATE SALT, SUCH AS A (D)(-) TARTRATE SALT OR A (LJ(+) TARTRATE SALT, A HYDROCHLORIDE SALT, A CITRATE SALT, A MALATE SALT, A FUMARATE SALT, A SUCCINATE SALT, A BENZOATE SALT, A BENZENESULFONATE SALT, A PAMOATE SALT, A FORMATE SALT, A MALONATE SALT, A 1,5- NAPHTHALENEDISULFONATE SALT, A SALICYLATE SALT, A CYCLOHEXANESULFAMATE SALT, A LACTATE SALT, A MANDELATE SALT, AQ GLUTARATE SALT, AN ADIPATE SALT, A SQUARATE SALT, A VANILLATE SALT, AN OXALOACETATE SALT, AN ASCORBATE SALT AND A SULFATE SALT. |