发明名称 |
POLYMORPHIC FORM OF A [1, 2, 4] TRIAZOLO [4, 3-A] PYRIDINE DERIVATIVE FOR TREATING INFLAMMATORY DISEASES |
摘要 |
Disclosed is a polymorphic form B of N-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1Hpyrazol- 5-yl]-N'-{ 2-[(3-{ 2-[(2-hydroxyethyl)sulfanyl]phenyl} [1,2,4]triazolo[4,3-a]pyridin-6 yl)sulfanyl]benzyl} . Also disclosed is the use of this form in the treatment of TNF or p38-mediated diseases e.g. chronic obstructive pulmonary disease and a process to prepare said form.
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申请公布号 |
NZ587094(A) |
申请公布日期 |
2011.07.29 |
申请号 |
NZ20090587094 |
申请日期 |
2009.01.28 |
申请人 |
PFIZER LIMITED |
发明人 |
BUTCHER, KENNETH, JOHN |
分类号 |
A61K31/437;A61P29/00;C07D471/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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