摘要 |
CRYSTALLINE SOLVATES AND COMPLEXES OF (IS) -1, 5-ANHYDRO-L-C (3- ( (PHENYL) METHYL) PHENYL) -D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETESAbstractThe present invention relates to physical crystal structures of a compound of the formula 1: wherein RI, R2, R2a, R3 and R4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures. No Suitable Figure |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
GOUGOUTAS, JACK, Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT, P.;BIEN, JEFFREY, T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN, ANTHONY;NIRSCHL, ALEXANDRA, A.;SINGH, JANAK;DIMARCO, JOHN, D. |