发明名称 CRYSTALLINE SOLVATES AND COMPLEXES OF (1S) -1, 5-ANHYDRO-1-C- (3- ( (PHENYL) METHYL) PHENYL) -D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 CRYSTALLINE SOLVATES AND COMPLEXES OF (IS) -1, 5-ANHYDRO-L-C (3- ( (PHENYL) METHYL) PHENYL) -D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETESAbstractThe present invention relates to physical crystal structures of a compound of the formula 1: wherein RI, R2, R2a, R3 and R4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures. No Suitable Figure
申请公布号 SG172741(A1) 申请公布日期 2011.07.28
申请号 SG20110047727 申请日期 2007.06.21
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 GOUGOUTAS, JACK, Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT, P.;BIEN, JEFFREY, T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN, ANTHONY;NIRSCHL, ALEXANDRA, A.;SINGH, JANAK;DIMARCO, JOHN, D.
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