发明名称 NOVEL INTERMEDIATE AND PROCESS FOR PREPARING ENTECAVIR USING SAME
摘要 The present invention relates to a novel, high-yield and low-cost method for preparing entecavir, [1-S-(1α,3α,4,&bgr;]-2-amino-1,9-dihydro-9-[4-hydroxy-3-(hydroxymethyl)-2-methylenecyclopentyl]-6H-purin-6-one, an antiviral agent, and novel intermediates used therein.
申请公布号 SG171963(A1) 申请公布日期 2011.07.28
申请号 SG20110040870 申请日期 2009.12.24
申请人 HANMI HOLDINGS CO., LTD. 发明人 LEE, JAEHEON;PARK, GHA-SEUNG;KIM, JIN HEE;LEE, JI EUN;PARK, CHUL HYUN;CHOI, TAE JIN;PARK, EUN-JU;KIM, CHEOL KYUNG;LIM, EUN JUNG;CHANG, YOUNG-KIL;LEE, GWAN SUN
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