发明名称 |
PROCESS FOR SYNTHESIS OF BIARYL OXAZOLIDINONE |
摘要 |
PROBLEM TO BE SOLVED: To provide a process for preparing biaryl oxazolidinones useful as anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents. SOLUTION: In the process, the biaryl oxazolidinones are synthesized by the exemplary reaction formula below in a solvent in the presence of a base and a palladium catalyst. COPYRIGHT: (C)2011,JPO&INPIT |
申请公布号 |
JP2011137007(A) |
申请公布日期 |
2011.07.14 |
申请号 |
JP20110021739 |
申请日期 |
2011.02.03 |
申请人 |
RIB-X PHARMACEUTICALS INC |
发明人 |
WU YUSHENG;CHEN SHILI;CHEN YI;HANSELMANN ROGER;LOU RONGLIANG;ZHOU JIACHENG |
分类号 |
C07D263/38;A61K31/422;A61K31/4245;A61K31/427;A61K31/433;A61K31/4439;A61K31/454;A61K31/4725;A61K31/496;A61P1/00;A61P1/04;A61P11/00;A61P29/00;A61P31/04;A61P31/10;A61P31/12;A61P33/00;A61P35/00;C07B61/00;C07D263/20;C07D413/06;C07D413/10;C07D413/12;C07D413/14;C07D417/10;C07D417/12;C07D417/14 |
主分类号 |
C07D263/38 |
代理机构 |
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代理人 |
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地址 |
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