发明名称 Thyazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase
摘要 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amine compounds are described, which are useful as LTA4 hydrolase (LTA4H) modulators. Such compounds may be used in pharmaceutical compositions and methods for modulation of LTA4H and for the treatment of disease states, disorders, and conditions mediated by LTA4 hydrolase activity.
申请公布号 US2011159563(A1) 申请公布日期 2011.06.30
申请号 US201113039017 申请日期 2011.03.02
申请人 JANSSEN PHARMACEUTICAL NV 发明人 BACANI GENESIS M.;BROGGINI DIEGO;CHEUNG EUGENE Y.;CHROVIAN CHRISTA C.;DENG XIAOHU;FOURIE ANNE M.;GOMEZ LAURENT;GRICE CHERYL A.;KEARNEY AARON M.;LANDRY-BAYLE ADRIENNE M.;LEE-DUTRA ALICE;LIANG JIMMY T.;LOCHNER SUSANNE;MANI NEELAKANDHA S.;SANTILLAN, JR. ALEJANDRO;SAPPEY KATHLEEN;SEPASSI KIA;TANIS VIRGINIA M.;WICKBOLDT ALVAH T.;WIENER JOHN J. M.;ZINSER HARTMUT
分类号 C12N9/99;C07D513/04 主分类号 C12N9/99
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