发明名称 SYNTHESIS AND USE OF VILDAGLIPTIN FOR THE PREPARATION OF PHARMACEUTICAL DOSAGE FORMS
摘要 The present invention relates the synthesis of vildagliptin in the presence of phase transfer catalysts; as well as the use of vildagliptin or its pharmaceutically acceptable salts for the preparation of solid oral dosage forms.
申请公布号 WO2011012322(A3) 申请公布日期 2011.06.30
申请号 WO2010EP04689 申请日期 2010.07.30
申请人 KRKA, D.D., NOVO MESTO;ZUPET, ROK;SMODIS, JANEZ;STROPNIK, TADEJ;ANDERLUH, MARKO;VRBINC, MIHA;VRECER, FRANC;PECAVAR, ANICA;KUKEC, SIMON 发明人 ZUPET, ROK;SMODIS, JANEZ;STROPNIK, TADEJ;ANDERLUH, MARKO;VRBINC, MIHA;VRECER, FRANC;PECAVAR, ANICA;KUKEC, SIMON
分类号 C07D207/16;A61K9/16;A61K31/4015 主分类号 C07D207/16
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