发明名称 |
NOVEL 3-HYDROXY-5-ARYLISOTHIAZOLE DERIVATIVE |
摘要 |
<p>Disclosed are a GPR40 activator having as an active ingredient a compound with a novel GPR40 agonist effect, a salt thereof, or a solvate of either; disclosed in particular are an insulin secretagogue, and a prophylactic and/or therapeutic agent for diabetes and obesity, etc., wherein said compound is represented by formula (I) (wherein n is 0-2, p is 0-4, j is 0-3, k is 0-2; ring A is an aryl group or a heterocyclic group optionally substituted by L; ring B is a benzene ring, a pyridine ring, or a pyrimidine ring; X is O, S, or -NR7-; R1 to R7 and L represent a specific group).</p> |
申请公布号 |
WO2011078371(A1) |
申请公布日期 |
2011.06.30 |
申请号 |
WO2010JP73464 |
申请日期 |
2010.12.24 |
申请人 |
MOCHIDA PHARMACEUTICAL CO.,LTD.;OKANO, AKIHIRO;KOSUGA, NAOTO;OHKOUCHI, MUNETAKA;HOTTA, DAIDO;MAKABE, MUNEYOSHI |
发明人 |
OKANO, AKIHIRO;KOSUGA, NAOTO;OHKOUCHI, MUNETAKA;HOTTA, DAIDO;MAKABE, MUNEYOSHI |
分类号 |
C07D275/02;A61K31/425;A61K31/427;A61K31/4439;A61K31/506;A61P3/10;C07D417/12;C07D417/14 |
主分类号 |
C07D275/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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