发明名称 SUBSTITUTED N-(1H-INDAZOL-4-YL)IMIDAZO[1, 2-A]PYRIDINE-3- CARBOXAMIDE COMPOUNDS AS CFMS INHIBITORS
摘要 <p>Compounds of Formula (I): and pharmaceutically acceptable salts thereof in which R1, R2, R3, R4 and R5 have the meanings given in the specification, are inhibitors of cFMS and are useful in the treatment of bone-related diseases, cancer, autoimmune disorders, inflammatory diseases, cardiovascular diseases and pain.</p>
申请公布号 WO2011079076(A1) 申请公布日期 2011.06.30
申请号 WO2010US61341 申请日期 2010.12.20
申请人 ARRAY BIOPHARMA INC.;BOYS, MARK LAURENCE;BRADLEY, MICHAEL;DELISLE, ROBERT KIRK;HENNINGS, D. DAVID;KENNEDY, APRIL L.;MARMSATER, FREDRIK P.;MEDINA, MATTHEW;MUNSON, MARK C.;RAST, BRYSON;RIZZI, JAMES P.;RODRIGUEZ, MARTHA E.;TOPALOV, GEORGE T.;ZHAO, QIAN 发明人 BOYS, MARK LAURENCE;BRADLEY, MICHAEL;DELISLE, ROBERT KIRK;HENNINGS, D. DAVID;KENNEDY, APRIL L.;MARMSATER, FREDRIK P.;MEDINA, MATTHEW;MUNSON, MARK C.;RAST, BRYSON;RIZZI, JAMES P.;RODRIGUEZ, MARTHA E.;TOPALOV, GEORGE T.;ZHAO, QIAN
分类号 C07D471/04;A61K31/437;A61K31/4985;A61P9/00;A61P19/08;A61P29/00;A61P35/00;C07D519/00 主分类号 C07D471/04
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