发明名称 |
SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS |
摘要 |
FIELD: medicine, pharmaceutics. ^ SUBSTANCE: invention refers to a compound of formula (I) or to its salt or ester in which radicals and symbols have the values presented in claim 1. These compounds are ACC inhibitors. ^ EFFECT: production of compounds to be applied as a therapeutic agent for various ACC-related disorders such as bacony liver, hyperlipidemia, obesity and diabetes. ^ 13 cl, 48 ex |
申请公布号 |
RU2422446(C2) |
申请公布日期 |
2011.06.27 |
申请号 |
RU20080106243 |
申请日期 |
2006.07.14 |
申请人 |
MERK SHARP EHND DOMEH KORP.;BANIU FARMAS'JUTIKAL KO., LTD. |
发明人 |
JAMAKAVA TAKERU;DZONA KHIDEKI;NIIJAMA KENDZI;JAMADA KODZI;IINO TOMOKHARU;OKHKUBO MITSURU;IMAMURA KHIDEAKI;KUSUNOKI DZUN;JANG LIKHU |
分类号 |
A61K31/438;A61P3/00;C07D491/107;C07D491/20 |
主分类号 |
A61K31/438 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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