发明名称 |
A PROCESS FOR PREPARATION OF ROSUVASTATIN ACETONIDE CALCIUM |
摘要 |
<p>The present invention is in relation to a process for preparation of HMG-CoA reductase inhibitor. More particularly, the present invention provides a process for preparation of (3R,5S,6E) 6-{2-[4-(4-Fluoro-phenyl)-6-isopropyl-2-(methanesulfonyl-methyl-amino)-pyrimidin-5-yl]-vinyl}-2,2-dimethyl-[1,3]dioxan-4-yl)-acetic acid, calcium salt (Rosuvastatin acetonide calcium) which is used for treating hypercholesterolemia.</p> |
申请公布号 |
EP2334667(A1) |
申请公布日期 |
2011.06.22 |
申请号 |
EP20080876921 |
申请日期 |
2008.10.22 |
申请人 |
BIOCON LIMITED |
发明人 |
SRINIVAS, PULLELA, VENKATA;ANEGONDI, SREENIVASA, PRASAD;RAJMAHENDRA, SHANMUGHASAMY;PONNUSAMY, THANGARASU |
分类号 |
C07D405/06;A61K31/075;A61K31/10;A61K31/357;A61K31/506;A61P7/00 |
主分类号 |
C07D405/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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