发明名称 A PROCESS FOR PREPARATION OF ROSUVASTATIN ACETONIDE CALCIUM
摘要 <p>The present invention is in relation to a process for preparation of HMG-CoA reductase inhibitor. More particularly, the present invention provides a process for preparation of (3R,5S,6E) 6-{2-[4-(4-Fluoro-phenyl)-6-isopropyl-2-(methanesulfonyl-methyl-amino)-pyrimidin-5-yl]-vinyl}-2,2-dimethyl-[1,3]dioxan-4-yl)-acetic acid, calcium salt (Rosuvastatin acetonide calcium) which is used for treating hypercholesterolemia.</p>
申请公布号 EP2334667(A1) 申请公布日期 2011.06.22
申请号 EP20080876921 申请日期 2008.10.22
申请人 BIOCON LIMITED 发明人 SRINIVAS, PULLELA, VENKATA;ANEGONDI, SREENIVASA, PRASAD;RAJMAHENDRA, SHANMUGHASAMY;PONNUSAMY, THANGARASU
分类号 C07D405/06;A61K31/075;A61K31/10;A61K31/357;A61K31/506;A61P7/00 主分类号 C07D405/06
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