发明名称 |
8-HYDROXYQUINOLINE DERIVATIVES FOR THE TREATMENT OF HEMATOLOGICAL MALIGNANCIES |
摘要 |
The application relates to compositions and methods for treating hematological malignancies and proliferative diseases, disorders and conditions involving increased D-cyclin expression. In particular, the application relates to compositions and methods for treating the hematological malignancies acute myeloid leukemia (AML), lymphoma and multiple myeloma (MM) using 5-nitrogen substituted hydroxy quinolones as well as 7-bromo-5-chloro substituted hydroxy quinolones and 5-chloro substituted hydroxy quinolones.
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申请公布号 |
US2011144155(A1) |
申请公布日期 |
2011.06.16 |
申请号 |
US20090995968 |
申请日期 |
2009.06.05 |
申请人 |
SCHIMMER AARON D;LI XIAOMING;BATEY ROBERT;WOOD TABITHA;MAO XINLIANG |
发明人 |
SCHIMMER AARON D.;LI XIAOMING;BATEY ROBERT;WOOD TABITHA;MAO XINLIANG |
分类号 |
A61K31/47;A61P35/02 |
主分类号 |
A61K31/47 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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