发明名称 5-HYDROXY-4-AMINOMETHYL-1-CYCLOHEXANE OR (CYCLOHEPTYL)--3-ALKOXYCARBONYL INDOLE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE ANTIVIRAL SALTS THEREOF AND A METHOD FOR THE PRODUCTION THEREOF
摘要 The invention relates to novel 5-hydroxy-4-aminomethyl-1-cyclohexane or (cycloheptyl)-3-alkoxycarbonyl indole derivatives of general formula (I) and to pharmaceutically acceptable salts thereof exhibiting antiviral activity and to a method for the production thereof. The compounds can be used for treating and/or preventing such viral diseases as pig and bird flu. The invention also relates to a method for producing the compounds of general formula (I), wherein X is hydrogen, chlorine or iodine, n=1 or 2, R3 is C1-C5 alkyl, Alk is a C1-C6 alkyl group, R1 and R2 are independently selected from C1-C4 alkyl, mainly methyl, or the NR1R2 group means groups of formula (II).
申请公布号 US2011144353(A1) 申请公布日期 2011.06.16
申请号 US20100950845 申请日期 2010.11.19
申请人 OBSCHESTVO S ORGANICHENNOY OTVETSTVENNOSTJU <<BINATEKH>> 发明人 VERKHOVSKY JURY G.;VERKHOVSKAYA N.;TSYSHKOVA NINA G.;ROZIEV RAKHIMDZHAN A.;TSYB ANATOLIY F.;GONCHAROVA ANNA YA.;TROFIMOV FEDOR A.;PODGORODNICHENKO VLADIMIR K.
分类号 C07D209/42 主分类号 C07D209/42
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