发明名称 SOLID STATE FORMS OF FESOTERODINE INTERMEDIATES
摘要 Provided herein are novel solid state forms of fesoterodine intermediates, (R)-4-benzyloxy-3-(3-diisopropylamino-1-phenylpropyl)-benzoic acid and (R)-[4-benzyloxy-3-(3-diisopropylamino-1-phenylpropyl)-phenyl]-methanol, and processes for their preparation thereof. The solid state intermediates are useful for preparing fesoterodine or a pharmaceutically acceptable salt thereof in high purity.
申请公布号 US2011124903(A1) 申请公布日期 2011.05.26
申请号 US20100949102 申请日期 2010.11.18
申请人 ACTAVIS GROUP PTC EHF 发明人 CHARUGUNDLA KISHORE;KUMAR UDHAYA;KUMAR NEELA PRAVEEN;PRADHAN NITIN SHARADCHANDRA
分类号 C07C69/017;C07C211/27 主分类号 C07C69/017
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