发明名称 |
DIAGNOSTIC AGENTS SELECTIVE AGAINST METALLOPROTEASES |
摘要 |
The invention relates to aryl-sulphonamido compounds endowed with affinity against metallo proteases MMP, having formula (I) below
wherein R, R 1 , R 2 , R 3 , G and n have the meanings reported in the specification, properly labelled with diagnostic imaging moieties or even radiotherapeutic moieties. The invention also refers to the process for their preparation, to pharmaceutical compositions comprising them and to their use as diagnostic imaging agents or radiotherapeutic agents. |
申请公布号 |
EP2320954(A1) |
申请公布日期 |
2011.05.18 |
申请号 |
EP20090800042 |
申请日期 |
2009.07.21 |
申请人 |
BRACCO IMAGING S.P.A |
发明人 |
ROSSELLO, ARMANDO;NUTI, ELISA;AVRAMOVA, STANISLAVA IVANOVA;UGGERI, FULVIO;MAIOCCHI, ALESSANDRO |
分类号 |
A61K49/00;A61K49/10;A61K49/22;A61K51/04;A61P43/00;C07C311/48;C07D295/08;C07D295/088 |
主分类号 |
A61K49/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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