发明名称 HETEROARYLAMINOQUINOLINES AS TGF-BETA RECEPTOR KINASE INHIBITORS
摘要 Novel hetarylaminoquinoline derivatives of formula (I) wherein X, Z, Het, R1, R2, R3 and R4 have the meaning according to claim 1, are inhibitors of ATP consuming proteins, and can be employed, inter alia, for the treatment of tumors.
申请公布号 WO2011054433(A1) 申请公布日期 2011.05.12
申请号 WO2010EP06239 申请日期 2010.10.12
申请人 MERCK PATENT GMBH;JONCZYK, ALFRED;AMENDT, CHRISTIANE;ZENKE, FRANK 发明人 JONCZYK, ALFRED;AMENDT, CHRISTIANE;ZENKE, FRANK
分类号 A61K31/4706;A61K31/4709;A61P35/00;C07D401/12;C07D401/14;C07D471/04 主分类号 A61K31/4706
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