发明名称 |
HETEROARYLAMINOQUINOLINES AS TGF-BETA RECEPTOR KINASE INHIBITORS |
摘要 |
Novel hetarylaminoquinoline derivatives of formula (I) wherein X, Z, Het, R1, R2, R3 and R4 have the meaning according to claim 1, are inhibitors of ATP consuming proteins, and can be employed, inter alia, for the treatment of tumors. |
申请公布号 |
WO2011054433(A1) |
申请公布日期 |
2011.05.12 |
申请号 |
WO2010EP06239 |
申请日期 |
2010.10.12 |
申请人 |
MERCK PATENT GMBH;JONCZYK, ALFRED;AMENDT, CHRISTIANE;ZENKE, FRANK |
发明人 |
JONCZYK, ALFRED;AMENDT, CHRISTIANE;ZENKE, FRANK |
分类号 |
A61K31/4706;A61K31/4709;A61P35/00;C07D401/12;C07D401/14;C07D471/04 |
主分类号 |
A61K31/4706 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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