发明名称 GPBP INHIBITION USING Q2 PEPTIDOMIMETICS
摘要 Disclosed are compounds of formula (I) that inhibiting GPBP activity, making them useful as therapeutics in antibody-mediated disorders, drug-resistant cancer, inflammation, protein misfolding and ER stress-mediated disorders, and aberrant apoptosis.
申请公布号 WO2011054530(A1) 申请公布日期 2011.05.12
申请号 WO2010EP06757 申请日期 2010.11.05
申请人 FIBROSTATIN, S.L.;SAUS, JUAN;FUSTERO, SANTOS;SANZ-CERVERA, F. JUAN;PEREZ-PAYA, ENRIQUE;BLASCO, RAUEL;REVERT-ROS, FRANCISCO;REVERT, FERNANDO 发明人 SAUS, JUAN;FUSTERO, SANTOS;SANZ-CERVERA, F. JUAN;PEREZ-PAYA, ENRIQUE;BLASCO, RAUEL;REVERT-ROS, FRANCISCO;REVERT, FERNANDO
分类号 C07C47/565;A61P29/00;A61P37/00;C07C45/68;C07C59/52;C07C59/56;C07C59/64;C07C67/343;C07C69/732;C07C69/734;C07C69/738;C07C309/65;C07D213/34;C07D213/48;C07D213/55 主分类号 C07C47/565
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