The present invention provides methods for preparing TLR-4 receptor agonist E6020:
and stereoisomers thereof, which compounds are useful as an immunological adjuvants when co-administered with antigens such as vaccines for bacterial and viral diseases. Also provided are synthetic intermediates.
申请公布号
EP2292628(A3)
申请公布日期
2011.05.11
申请号
EP20100012396
申请日期
2006.06.30
申请人
EISAI R&D MANAGEMENT CO., LTD.
发明人
FANG, FRANCIS G.;FOY, JAMES E.;HAWKINS, LYNN;LEMELIN, CHARLES;LESCARBEAU, ANDRE;NIU, XIANG;WU, KUO-MING