发明名称 HETEROCYCLYL SUBSTITUTED ARYLINDENOPY-RIMIDINES AND THEIR USE AS HIGHLY SELECTIVE ADENOSINE A2A RECEPTOR ANTAGONISTS
摘要 <p>This invention relates to a novel arylindenopyrimidine, A, and its therapeutic and prophylactic uses. Disorders treated and/or prevented include Parkinson's Disease. Formula (I) wherein X. R2, R3, and R4 are as defined in the specification.</p>
申请公布号 WO2011053510(A1) 申请公布日期 2011.05.05
申请号 WO2010US53590 申请日期 2010.10.21
申请人 JANSSEN PHARMACEUTICA NV;JACKSON, PAUL, F.;POWELL, MARK;SHOOK, BRIAN, CHRISTOPHER;WANG, AIHUA 发明人 JACKSON, PAUL, F.;POWELL, MARK;SHOOK, BRIAN, CHRISTOPHER;WANG, AIHUA
分类号 C07D239/70;A61K31/519;A61P25/00;A61P25/16;A61P25/22;A61P25/24;A61P25/28;A61P25/30;C07D401/12 主分类号 C07D239/70
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