发明名称 |
PROCESS FOR PREPARING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR |
摘要 |
<p>The present invention relates to processes for preparing solid state forms of N-(4-(7-azabicyclo[2.2. 1]heptan-7-yl)-2-(trifluoromethyl)phenyl)-4-oxo-5-(trifluoromethyl)-1,4-dihydroquinoline-3-carboxamide, including Compound 1 Form A, Compound 1 Form A- HCl, Compound 1 Form B, and Compound 1 Form B-HCl, any combination of these forms, pharmaceutical compositions thereof, and methods of treatment therewith.</p> |
申请公布号 |
CA2778492(A1) |
申请公布日期 |
2011.04.28 |
申请号 |
CA20102778492 |
申请日期 |
2010.10.21 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
AMBHAIKAR, NARENDRA BHALCHANDRA;HUGHES, ROBERT;HURLEY, DENNIS JAMES;LEE, ELAINE CHUNGMIN;LITTLER, BENJAMIN;NUMA, MEHDI;ROEPER, STEFANIE;SHETH, URVI |
分类号 |
C07D215/56;C07D487/08 |
主分类号 |
C07D215/56 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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