发明名称 |
PARTICLES COMPRISING A SALT OF 8-HYDROXY-2-[[(1R)-2-(4-METHOXYPHENYL)-1-METHYLETHYL]AMINO]ETHYL]-2(1H)-QUINOLINONE HAVING IMPROVED ADHESION PROPERTIES FOR POWDER FORMULATIONS FOR INHALATION |
摘要 |
Powder particles comprising a pharmaceutically acceptable salt of 8-hydroxy-5-[(1R)-1-hydroxy-2-[[(1R)-2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]-2(1H)-quinolinone (carmoterol) having a specific properties exhibit improved adhesion properties for dry powder formulations for inhalation. Such particles are useful for formulations in the form of powders for inhalation and the treatment of certain conditions and diseases.
|
申请公布号 |
US2011097409(A1) |
申请公布日期 |
2011.04.28 |
申请号 |
US20090625758 |
申请日期 |
2009.11.25 |
申请人 |
CHIESI FARMACEUTICI S.P.A. |
发明人 |
BUTTINI FRANCESCA;COLOMBO PAOLO;PARLATI CHIARA;COCCONI DANIELA;MUSA ROSSELLA |
分类号 |
A61K9/14;A61K31/4704;A61K31/56;A61K31/58;A61P11/00;B29B9/12;C07D215/26 |
主分类号 |
A61K9/14 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|